Jean-Michel Chezal

Affiliations

Inserm, Imagerie Moléculaire et Stratégies Théranostiques, UMR 1240, Université Clermont Auvergne, F-63000 Clermont-Ferrand, France.

Publications (15)

A Convenient Route to New (Radio)Fluorinated and (Radio)Iodinated Cyclic Tyrosine Analogs.

Pharmaceuticals (Basel, Switzerland)

Avec: Maria Noelia Chao , Eric Debiton , Damien Canitrot , Tiffany Witkowski , Sophie Levesque , Françoise Degoul , Sébastien Tarrit , Barbara Wenzel , Elisabeth Miot-Noirault , Audrey Serre , Aurélie Maisonial-Besset

Optimization of IEDDA bioorthogonal system: Efficient process to improve trans-cyclooctene/tetrazine interaction.

European journal of medicinal chemistry

Avec: Jean-Baptiste Béquignat , Nancy Ty , Aurélie Rondon , Ludivine Taiariol , Françoise Degoul , Damien Canitrot , Mercedes Quintana , Isabelle Navarro-Teulon , Elisabeth Miot-Noirault , Claude Boucheix , Emmanuel Moreau

Design, synthesis and evaluation of targeted hypoxia-activated prodrugs applied to chondrosarcoma chemotherapy.

Bioorganic chemistry

Avec: Yvain Gerard , Aurélien Voissière , Caroline Peyrode , Marie-Josephe Galmier , Elise Maubert , Donia Ghedira , Sebastien Tarrit , Vincent Gaumet , Damien Canitrot , Elisabeth Miot-Noirault , Valérie Weber

Synthesis and

Journal of materials chemistry. B

Avec: Axel Cordonnier , Damien Boyer , Sophie Besse , Rodolphe Valleix , Rachid Mahiou , Mercedes Quintana , Arnaud Briat , Mhammed Benbakkar , Frédérique Penault-Llorca , Aurélie Maisonial-Besset , Benoit Maunit , Sébastien Tarrit , Magali Vivier , Tiffany Witkowski , Leslie Mazuel , Françoise Degoul , Elisabeth Miot-Noirault ,

Targeted Radionuclide Therapy Decreases Melanoma Lung Invasion by Modifying Epithelial-Mesenchymal Transition-Like Mechanisms.

Translational oncology

Avec: Hussein Akil , Jacques Rouanet , Claire Viallard , Sophie Besse , Philippe Auzeloux , Elisabeth Miot-Noirault , Mercedes Quintana , Françoise Degoul

Targeting cyclic nucleotide phosphodiesterase 5 (PDE5) in brain: Toward the development of a PET radioligand labeled with fluorine-18.

Bioorganic chemistry

Avec: Barbara Wenzel , Jianrong Liu , Sladjana Dukic-Stefanovic , Winnie Deuther-Conrad , Rodrigo Teodoro , Friedrich-Alexander Ludwig , Emmanuel Moreau , Peter Brust , Aurelie Maisonial-Besset

Improved automated one-pot two-step radiosynthesis of (S)-[

EJNMMI radiopharmacy and chemistry

Avec: Aurélie Maisonial-Besset , David Kryza , Klaus Kopka , Sophie Levesque , Emmanuel Moreau , Barbara Wenzel ,

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EJNMMI research

Avec: Elodie Jouberton , Sébastien Schmitt , Emmanuel Chautard , Aurélie Maisonial-Besset , Marie Roy , Nina Radosevic-Robin , Elisabeth Miot-Noirault , Yann Bouvet , Florent Cachin

Relevance of the combination of external beam radiotherapy with the hypoxia-activated prodrug ICF05016 in an experimental model of extraskeletal myxoid chondrosarcoma.

Investigational new drugs

Avec: Elise Maubert , Valérie Weber , Aurélien Voissière , Yvain Gérard , Véronique Dedieu , Françoise Degoul , Emmanuel Chautard , Elisabeth Miot-Noirault

Phase I study of [

BMC cancer

Avec: Emilie Thivat , Jacques Rouanet , Philippe Auzeloux , Nicolas Sas , Elodie Jouberton , Sophie Levesque , Tommy Billoux , Sandrine Mansard , Ioana Molnar , Marion Chanchou , Giovanna Fois , Lydia Maigne , Elisabeth Miot-Noirault , Michel D'Incan , Xavier Durando , Florent Cachin

Novel Radioiodinated and Radiofluorinated Analogues of FT-2102 for SPECT or PET Imaging of mIDH1 Mutant Tumours.

Molecules (Basel, Switzerland)

Avec: Valérie Weber , Lucie Arnaud , Sladjana Dukic-Stefanovic , Barbara Wenzel , Valérie Roux , Thu-Hang Lai , Rodrigo Teodoro , Klaus Kopka , Elisabeth Miot-Noirault , Winnie Deuther-Conrad , Aurélie Maisonial-Besset

Branched pegylated linker-auristatin to control hydrophobicity for the production of homogeneous minibody-drug conjugate against HER2-positive breast cancer.

Journal of controlled release : official journal of the Controlled Release Society

Avec: Emmanuel Douez , Emilie Allard-Vannier , Imène Ait Mohamed Amar , Louis Jolivet , Fanny Boursin , Aurélie Maisonial-Besset , Tiffany Witkowski , Cyril Colas , Stéphanie Letast , Etienne Auvert , Caroline Denevault-Sabourin , Nicolas Aubrey , Nicolas Joubert

Synthesis and In Vitro Comparison of DOTA, NODAGA and 15-5 Macrocycles as Chelators for the

Molecules (Basel, Switzerland)

Avec: Aurélie Maisonial-Besset , Tiffany Witkowski , Mercedes Quintana , Sophie Besse , Vincent Gaumet , Axel Cordonnier , Cyrille Alliot , Aurélien Vidal , Caroline Denevault-Sabourin , Sébastien Tarrit , Sophie Levesque , Elisabeth Miot-Noirault ,

Homologation of the Alkyl Side Chain of Antimitotic Phenyl 4-(2-Oxo-3-alkylimidazolidin-1-yl)benzenesulfonate Prodrugs Selectively Targeting CYP1A1-Expressing Breast Cancers Improves Their Stability in Rodent Liver Microsomes.

Journal of medicinal chemistry

Avec: Atziri Corin Chavez Alvarez , Chahrazed Bouzriba , Emmanuel Moreau , Philippe Auzeloux , Sophie Besse , Vincent Ouellette , Mitra Zarifi Khosroshahi , Marie-France Côté , Sylvie Pilote , Elisabeth Miot-Noirault , Chantale Simard , René C-Gaudreault , Sébastien Fortin

From netrin-1-targeted SPECT/CT to internal radiotherapy for management of advanced solid tumors.

EMBO molecular medicine

Avec: David Kryza , Jennifer Wischhusen , Mathieu Richaud , Maëva Hervieu , Jacqueline Sidi Boumedine , Jean-Guy Delcros , Sophie Besse , Thomas Baudier , Pierre-Alexandre Laval , Silvia Breusa , Erwan Boutault , Hugo Clermidy , Nicolas Rama , Benjamin Ducarouge , Mojgan Devouassoux-Shisheboran , Anne-Laure Giraudet , Thomas Walter , Patrick Mehlen , David Sarrut , Benjamin Gibert

Réseau de co-auteurs

Elisabeth Miot-Noirault 11 collaborations

Aurélie Maisonial-Besset 7 collaborations

Françoise Degoul 5 collaborations

Sophie Besse 5 collaborations

Tiffany Witkowski 4 collaborations

Sophie Levesque 4 collaborations

Barbara Wenzel 4 collaborations

Mercedes Quintana 4 collaborations

Emmanuel Moreau 4 collaborations

Damien Canitrot 3 collaborations

Sébastien Tarrit 3 collaborations

Valérie Weber 3 collaborations

Philippe Auzeloux 3 collaborations

Aurélien Voissière 2 collaborations

Elise Maubert 2 collaborations

Vincent Gaumet 2 collaborations

Axel Cordonnier 2 collaborations

Jacques Rouanet 2 collaborations

Sladjana Dukic-Stefanovic 2 collaborations

Winnie Deuther-Conrad 2 collaborations

Rodrigo Teodoro 2 collaborations

David Kryza 2 collaborations

Klaus Kopka 2 collaborations

Elodie Jouberton 2 collaborations

Emmanuel Chautard 2 collaborations

Florent Cachin 2 collaborations

Caroline Denevault-Sabourin 2 collaborations

Maria Noelia Chao 1 collaboration

Eric Debiton 1 collaboration

Audrey Serre 1 collaboration

Jean-Baptiste Béquignat 1 collaboration

Nancy Ty 1 collaboration

Aurélie Rondon 1 collaboration

Ludivine Taiariol 1 collaboration

Isabelle Navarro-Teulon 1 collaboration

Claude Boucheix 1 collaboration

Yvain Gerard 1 collaboration

Caroline Peyrode 1 collaboration

Marie-Josephe Galmier 1 collaboration

Donia Ghedira 1 collaboration

Sebastien Tarrit 1 collaboration

Damien Boyer 1 collaboration

Rodolphe Valleix 1 collaboration

Rachid Mahiou 1 collaboration

Arnaud Briat 1 collaboration

Mhammed Benbakkar 1 collaboration

Frédérique Penault-Llorca 1 collaboration

Benoit Maunit 1 collaboration

Magali Vivier 1 collaboration

Leslie Mazuel 1 collaboration

Hussein Akil 1 collaboration

Claire Viallard 1 collaboration

Jianrong Liu 1 collaboration

Friedrich-Alexander Ludwig 1 collaboration

Peter Brust 1 collaboration

Aurelie Maisonial-Besset 1 collaboration

Sébastien Schmitt 1 collaboration

Marie Roy 1 collaboration

Nina Radosevic-Robin 1 collaboration

Yann Bouvet 1 collaboration

Yvain Gérard 1 collaboration

Véronique Dedieu 1 collaboration

Emilie Thivat 1 collaboration

Nicolas Sas 1 collaboration

Tommy Billoux 1 collaboration

Sandrine Mansard 1 collaboration

Ioana Molnar 1 collaboration

Marion Chanchou 1 collaboration

Giovanna Fois 1 collaboration

Lydia Maigne 1 collaboration

Michel D'Incan 1 collaboration

Xavier Durando 1 collaboration

Lucie Arnaud 1 collaboration

Valérie Roux 1 collaboration

Thu-Hang Lai 1 collaboration

Emmanuel Douez 1 collaboration

Emilie Allard-Vannier 1 collaboration

Imène Ait Mohamed Amar 1 collaboration

Louis Jolivet 1 collaboration

Fanny Boursin 1 collaboration

Cyril Colas 1 collaboration

Stéphanie Letast 1 collaboration

Etienne Auvert 1 collaboration

Nicolas Aubrey 1 collaboration

Nicolas Joubert 1 collaboration

Cyrille Alliot 1 collaboration

Aurélien Vidal 1 collaboration

Atziri Corin Chavez Alvarez 1 collaboration

Chahrazed Bouzriba 1 collaboration

Vincent Ouellette 1 collaboration

Mitra Zarifi Khosroshahi 1 collaboration

Marie-France Côté 1 collaboration

Sylvie Pilote 1 collaboration

Chantale Simard 1 collaboration

René C-Gaudreault 1 collaboration

Sébastien Fortin 1 collaboration

Jennifer Wischhusen 1 collaboration

Mathieu Richaud 1 collaboration

Maëva Hervieu 1 collaboration

Jacqueline Sidi Boumedine 1 collaboration

Jean-Guy Delcros 1 collaboration

Thomas Baudier 1 collaboration

Pierre-Alexandre Laval 1 collaboration

Silvia Breusa 1 collaboration

Erwan Boutault 1 collaboration

Hugo Clermidy 1 collaboration

Nicolas Rama 1 collaboration

Benjamin Ducarouge 1 collaboration

Mojgan Devouassoux-Shisheboran 1 collaboration

Anne-Laure Giraudet 1 collaboration

Thomas Walter 1 collaboration

Patrick Mehlen 1 collaboration

David Sarrut 1 collaboration

Benjamin Gibert 1 collaboration