Barbara Malawska

Affiliations
  • Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland.
ORCID: 0000-0003-4637-5820

Publications (26)

Dual Inhibitors of Amyloid-β and Tau Aggregation with Amyloid-β Disaggregating Properties: Extended

ACS chemical neuroscience
Avec: Anna Pasieka , Dawid Panek , Natalia Szałaj , Alba Espargaró , Anna Więckowska , Raimon Sabaté , Marek Bajda

Novel Functionalized Amino Acids as Inhibitors of GABA Transporters with Analgesic Activity.

ACS chemical neuroscience
Avec: Beata Gryzło , Paula Zaręba , Katarzyna Malawska , Gabriela Mazur , Anna Rapacz , Kamil Ła Tka , Georg C Höfner , Gniewomir Latacz , Marek Bajda , Kinga Sałat , Klaus T Wanner , Katarzyna Kulig

Cyanobiphenyls: Novel H

Bioorganic chemistry
Avec: Justyna Godyń , Paula Zaręba , Dorota Łażewska , Dorota Stary , David Reiner-Link , Annika Frank , Gniewomir Latacz , Szczepan Mogilski , Maria Kaleta , Agata Doroz-Płonka , Annamaria Lubelska , Ewelina Honkisz-Orzechowska , Agnieszka Olejarz-Maciej , Jadwiga Handzlik , Holger Stark , Katarzyna Kieć-Kononowicz , Marek Bajda

Discovery of new, highly potent and selective inhibitors of BuChE - design, synthesis, in vitro and in vivo evaluation and crystallography studies.

European journal of medicinal chemistry
Avec: Dawid Panek , Anna Pasieka , Gniewomir Latacz , Paula Zaręba , Michał Szczęch , Justyna Godyń , Fabien Chantegreil , Florian Nachon , Xavier Brazzolotto , Anna Skrzypczak-Wiercioch , Maria Walczak , Magdalena Smolik , Kinga Sałat , Georg Höfner , Klaus Wanner , Anna Więckowska ,

Search for new multi-target compounds against Alzheimer's disease among histamine H

European journal of medicinal chemistry
Avec: Marek Bajda , Dorota Łażewska , Justyna Godyń , Paula Zaręba , Kamil Kuder , Stefanie Hagenow , Kamil Łątka , Ewelina Stawarska , Holger Stark , Katarzyna Kieć-Kononowicz ,

Discovery of 1-(phenylsulfonyl)-1H-indole-based multifunctional ligands targeting cholinesterases and 5-HT

European journal of medicinal chemistry
Avec: Tomasz Wichur , Anna Pasieka , Justyna Godyń , Dawid Panek , Izabella Góral , Gniewomir Latacz , Ewelina Honkisz-Orzechowska , Adam Bucki , Agata Siwek , Monika Głuch-Lutwin , Damijan Knez , Xavier Brazzolotto , Stanislav Gobec , Marcin Kołaczkowski , Raimon Sabate , Anna Więckowska

1-Benzylpyrrolidine-3-amine-based BuChE inhibitors with anti-aggregating, antioxidant and metal-chelating properties as multifunctional agents against Alzheimer's disease.

European journal of medicinal chemistry
Avec: Tomasz Wichur , Anna Więckowska , Krzysztof Więckowski , Justyna Godyń , Jakub Jończyk , Álvaro Del Río Valdivieso , Dawid Panek , Anna Pasieka , Raimon Sabaté , Damijan Knez , Stanislav Gobec ,

A walk through tau therapeutic strategies.

Acta neuropathologica communications
Avec: Santosh Jadhav , Jesus Avila , Michael Schöll , Gabor G Kovacs , Enikö Kövari , Rostislav Skrabana , Lewis D Evans , Eva Kontsekova , Rohan de Silva , Luc Buee , Norbert Zilka

Novel application of capillary electrophoresis with a liposome coated capillary for prediction of blood-brain barrier permeability.

Talanta
Avec: Justyna Godyń , Dominika Gucwa , Tereza Kobrlova , Martin Novak , Ondrej Soukup , Marek Bajda

Dual Action of Dipyridothiazine and Quinobenzothiazine Derivatives-Anticancer and Cholinesterase-Inhibiting Activity.

Molecules (Basel, Switzerland)
Avec: Jakub Jończyk , Justyna Godyń , Ewelina Stawarska , Beata Morak-Młodawska , Małgorzata Jeleń , Krystian Pluta ,

Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT

European journal of medicinal chemistry
Avec: Tomasz Wichur , Justyna Godyń , Izabella Góral , Gniewomir Latacz , Adam Bucki , Agata Siwek , Monika Głuch-Lutwin , Barbara Mordyl , Joanna Śniecikowska , Maria Walczak , Damijan Knez , Marko Jukič , Kinga Sałat , Stanislav Gobec , Marcin Kołaczkowski , Xavier Brazzolotto , Anna Więckowska

Benzophenone Derivatives with Histamine H

Molecules (Basel, Switzerland)
Avec: Justyna Godyń , Paula Zaręba , Dorota Stary , Maria Kaleta , Kamil J Kuder , Gniewomir Latacz , Szczepan Mogilski , David Reiner-Link , Annika Frank , Agata Doroz-Płonka , Agnieszka Olejarz-Maciej , Sylwia Sudoł-Tałaj , Tobias Nolte , Jadwiga Handzlik , Holger Stark , Anna Więckowska , Katarzyna Kieć-Kononowicz , Dorota Łażewska , Marek Bajda

Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, β-secretase, and amyloid β aggregation as potential treatment of Alzheimer's disease.

European journal of medicinal chemistry
Avec: Paula Zaręba , Kamil Łątka , Gabriela Mazur , Beata Gryzło , Anna Pasieka , Justyna Godyń , Dawid Panek , Anna Skrzypczak-Wiercioch , Georg C Höfner , Gniewomir Latacz , Maciej Maj , Alba Espargaró , Raimon Sabaté , Krzysztof Jóźwiak , Klaus T Wanner , Kinga Sałat , Katarzyna Kulig , Marek Bajda

Novel mouse GABA uptake inhibitors with enhanced inhibitory activity toward mGAT3/4 and their effect on pain threshold in mice.

European journal of medicinal chemistry
Avec: Paula Zaręba , Beata Gryzło , Katarzyna Malawska , Kinga Sałat , Georg C Höfner , Alicja Nowaczyk , Łukasz Fijałkowski , Anna Rapacz , Adrian Podkowa , Anna Furgała , Paweł Żmudzki , Klaus T Wanner , Katarzyna Kulig

Development, Recent Achievements and Current Directions of Research into GABA Uptake Inhibitors.

Current medicinal chemistry
Avec: Paula Zaręba , Beata Gryzło , Gabriela Mazur ,

New Dual Small Molecules for Alzheimer's Disease Therapy Combining Histamine H

Journal of medicinal chemistry
Avec: Rim Malek , Raquel L Arribas , Alejandra Palomino-Antolin , Perle Totoson , Celine Demougeot , Tereza Kobrlova , Ondrej Soukup , Isabel Iriepa , Ignacio Moraleda , Daniel Diez-Iriepa , Justyna Godyń , Dawid Panek , Monika Głuch-Lutwin , Barbara Mordyl , Agata Siwek , Fakher Chabchoub , José Marco-Contelles , Katarzyna Kiec-Kononowicz , Javier Egea , Cristóbal de Los Ríos , Lhassane Ismaili

Pyridinium-2-carbaldoximes with quinolinium carboxamide moiety are simultaneous reactivators of acetylcholinesterase and butyrylcholinesterase inhibited by nerve agent surrogates.

Journal of enzyme inhibition and medicinal chemistry
Avec: Hyun Myung Lee , Rudolf Andrys , Jakub Jonczyk , Kyuneun Kim , Avinash G Vishakantegowda , David Malinak , Adam Skarka , Monika Schmidt , Michaela Vaskova , Kamil Latka , Marek Bajda , Young-Sik Jung , Kamil Musilek

Molecular Modeling Studies on the Multistep Reactivation Process of Organophosphate-Inhibited Acetylcholinesterase and Butyrylcholinesterase.

Biomolecules
Avec: Jakub Jończyk , Jędrzej Kukułowicz , Kamil Łątka , Young-Sik Jung , Kamil Musilek , Marek Bajda

Guanidines: Synthesis of Novel Histamine H

Pharmaceuticals (Basel, Switzerland)
Avec: Marek Staszewski , Magdalena Iwan , Tobias Werner , Marek Bajda , Justyna Godyń , Gniewomir Latacz , Agnieszka Korga-Plewko , Joanna Kubik , Natalia Szałaj , Holger Stark , Anna Więckowska , Krzysztof Walczyński

Multidirectional

Journal of enzyme inhibition and medicinal chemistry
Avec: Natalia Szałaj , Justyna Godyń , Jakub Jończyk , Anna Pasieka , Dawid Panek , Tomasz Wichur , Krzysztof Więckowski , Paula Zaręba , Marek Bajda , Anja Pislar , Raimon Sabate , Anna Więckowska

Discovery of multifunctional anti-Alzheimer's agents with a unique mechanism of action including inhibition of the enzyme butyrylcholinesterase and γ-aminobutyric acid transporters.

European journal of medicinal chemistry
Avec: Anna Pasieka , Dawid Panek , Jakub Jończyk , Justyna Godyń , Natalia Szałaj , Gniewomir Latacz , Julia Tabor , Eva Mezeiova , Fabien Chantegreil , José Dias , Damijan Knez , Junfeng Lu , Rongbiao Pi , Jan Korabecny , Xavier Brazzolotto , Stanislav Gobec , Georg Höfner , Klaus Wanner , Anna Więckowska ,

Search for multifunctional agents against Alzheimer's disease among non-imidazole histamine H3 receptor ligands. In vitro and in vivo pharmacological evaluation and computational studies of piperazine derivatives.

Bioorganic chemistry
Avec: Jakub Jończyk , Krzysztof Lodarski , Marek Staszewski , Justyna Godyń , Paula Zaręba , Ondrej Soukup , Jana Janockova , Jan Korabecny , Kinga Sałat , Natalia Malikowska-Racia , Michalina Hebda , Natalia Szałaj , Barbara Filipek , Krzysztof Walczyński , Marek Bajda

Rational design of new multitarget histamine H

European journal of medicinal chemistry
Avec: Dorota Łażewska , Marek Bajda , Maria Kaleta , Paula Zaręba , Agata Doroz-Płonka , Agata Siwek , Alaa Alachkar , Szczepan Mogilski , Ali Saad , Kamil Kuder , Agnieszka Olejarz-Maciej , Justyna Godyń , Dorota Stary , Sylwia Sudoł , Małgorzata Więcek , Gniewomir Latacz , Maria Walczak , Jadwiga Handzlik , Bassem Sadek , Katarzyna Kieć-Kononowicz

Biphenylalkoxyamine Derivatives-Histamine H

Molecules (Basel, Switzerland)
Avec: Dorota Łażewska , Paula Zaręba , Justyna Godyń , Agata Doroz-Płonka , Annika Frank , David Reiner-Link , Marek Bajda , Dorota Stary , Szczepan Mogilski , Agnieszka Olejarz-Maciej , Maria Kaleta , Holger Stark , Katarzyna Kieć-Kononowicz

Development of tricyclic N-benzyl-4-hydroxybutanamide derivatives as inhibitors of GABA transporters mGAT1-4 with anticonvulsant, antinociceptive, and antidepressant activity.

European journal of medicinal chemistry
Avec: Paula Zaręba , Kinga Sałat , Georg C Höfner , Kamil Łątka , Marek Bajda , Gniewomir Latacz , Krzysztof Kotniewicz , Anna Rapacz , Adrian Podkowa , Maciej Maj , Krzysztof Jóźwiak , Barbara Filipek , Klaus T Wanner , Katarzyna Kulig

Novel drug-like fluorenyl derivatives as selective butyrylcholinesterase and β-amyloid inhibitors for the treatment of Alzheimer's disease.

Bioorganic & medicinal chemistry
Avec: Anna Pasieka , Dawid Panek , Paula Zaręba , Emilia Sługocka , Natalia Gucwa , Alba Espargaró , Gniewomir Latacz , Nadia Khan , Adam Bucki , Raimon Sabaté , Anna Więckowska ,

Réseau de co-auteurs

Justyna Godyń 17 collaborations
Marek Bajda 15 collaborations
Paula Zaręba 14 collaborations
Gniewomir Latacz 12 collaborations
Anna Więckowska 10 collaborations
Dawid Panek 9 collaborations
Anna Pasieka 8 collaborations
Kinga Sałat 7 collaborations
Jakub Jończyk 6 collaborations
Natalia Szałaj 5 collaborations
Dorota Łażewska 5 collaborations
Holger Stark 5 collaborations
Katarzyna Kieć-Kononowicz 5 collaborations
Raimon Sabaté 4 collaborations
Beata Gryzło 4 collaborations
Georg C Höfner 4 collaborations
Klaus T Wanner 4 collaborations
Katarzyna Kulig 4 collaborations
Dorota Stary 4 collaborations
Szczepan Mogilski 4 collaborations
Maria Kaleta 4 collaborations
Agata Doroz-Płonka 4 collaborations
Agnieszka Olejarz-Maciej 4 collaborations
Xavier Brazzolotto 4 collaborations
Kamil Łątka 4 collaborations
Tomasz Wichur 4 collaborations
Agata Siwek 4 collaborations
Damijan Knez 4 collaborations
Stanislav Gobec 4 collaborations
Alba Espargaró 3 collaborations
Gabriela Mazur 3 collaborations
Anna Rapacz 3 collaborations
David Reiner-Link 3 collaborations
Annika Frank 3 collaborations
Jadwiga Handzlik 3 collaborations
Maria Walczak 3 collaborations
Adam Bucki 3 collaborations
Monika Głuch-Lutwin 3 collaborations
Ondrej Soukup 3 collaborations
Katarzyna Malawska 2 collaborations
Ewelina Honkisz-Orzechowska 2 collaborations
Fabien Chantegreil 2 collaborations
Anna Skrzypczak-Wiercioch 2 collaborations
Georg Höfner 2 collaborations
Klaus Wanner 2 collaborations
Kamil Kuder 2 collaborations
Ewelina Stawarska 2 collaborations
Izabella Góral 2 collaborations
Marcin Kołaczkowski 2 collaborations
Raimon Sabate 2 collaborations
Krzysztof Więckowski 2 collaborations
Tereza Kobrlova 2 collaborations
Barbara Mordyl 2 collaborations
Maciej Maj 2 collaborations
Krzysztof Jóźwiak 2 collaborations
Adrian Podkowa 2 collaborations
Young-Sik Jung 2 collaborations
Kamil Musilek 2 collaborations
Marek Staszewski 2 collaborations
Krzysztof Walczyński 2 collaborations
Jan Korabecny 2 collaborations
Barbara Filipek 2 collaborations
Kamil Ła Tka 1 collaboration
Annamaria Lubelska 1 collaboration
Michał Szczęch 1 collaboration
Florian Nachon 1 collaboration
Magdalena Smolik 1 collaboration
Stefanie Hagenow 1 collaboration
Álvaro Del Río Valdivieso 1 collaboration
Santosh Jadhav 1 collaboration
Jesus Avila 1 collaboration
Michael Schöll 1 collaboration
Gabor G Kovacs 1 collaboration
Enikö Kövari 1 collaboration
Rostislav Skrabana 1 collaboration
Lewis D Evans 1 collaboration
Eva Kontsekova 1 collaboration
Rohan de Silva 1 collaboration
Luc Buee 1 collaboration
Norbert Zilka 1 collaboration
Dominika Gucwa 1 collaboration
Martin Novak 1 collaboration
Beata Morak-Młodawska 1 collaboration
Małgorzata Jeleń 1 collaboration
Krystian Pluta 1 collaboration
Joanna Śniecikowska 1 collaboration
Marko Jukič 1 collaboration
Kamil J Kuder 1 collaboration
Sylwia Sudoł-Tałaj 1 collaboration
Tobias Nolte 1 collaboration
Alicja Nowaczyk 1 collaboration
Łukasz Fijałkowski 1 collaboration
Anna Furgała 1 collaboration
Paweł Żmudzki 1 collaboration
Rim Malek 1 collaboration
Raquel L Arribas 1 collaboration
Alejandra Palomino-Antolin 1 collaboration
Perle Totoson 1 collaboration
Celine Demougeot 1 collaboration
Isabel Iriepa 1 collaboration
Ignacio Moraleda 1 collaboration
Daniel Diez-Iriepa 1 collaboration
Fakher Chabchoub 1 collaboration
José Marco-Contelles 1 collaboration
Katarzyna Kiec-Kononowicz 1 collaboration
Javier Egea 1 collaboration
Cristóbal de Los Ríos 1 collaboration
Lhassane Ismaili 1 collaboration
Hyun Myung Lee 1 collaboration
Rudolf Andrys 1 collaboration
Jakub Jonczyk 1 collaboration
Kyuneun Kim 1 collaboration
Avinash G Vishakantegowda 1 collaboration
David Malinak 1 collaboration
Adam Skarka 1 collaboration
Monika Schmidt 1 collaboration
Michaela Vaskova 1 collaboration
Kamil Latka 1 collaboration
Jędrzej Kukułowicz 1 collaboration
Magdalena Iwan 1 collaboration
Tobias Werner 1 collaboration
Agnieszka Korga-Plewko 1 collaboration
Joanna Kubik 1 collaboration
Anja Pislar 1 collaboration
Julia Tabor 1 collaboration
Eva Mezeiova 1 collaboration
José Dias 1 collaboration
Junfeng Lu 1 collaboration
Rongbiao Pi 1 collaboration
Krzysztof Lodarski 1 collaboration
Jana Janockova 1 collaboration
Natalia Malikowska-Racia 1 collaboration
Michalina Hebda 1 collaboration
Alaa Alachkar 1 collaboration
Ali Saad 1 collaboration
Sylwia Sudoł 1 collaboration
Małgorzata Więcek 1 collaboration
Bassem Sadek 1 collaboration
Krzysztof Kotniewicz 1 collaboration
Emilia Sługocka 1 collaboration
Natalia Gucwa 1 collaboration
Nadia Khan 1 collaboration