Biological Evaluation of Noscapine analogues as Potent and Microtubule-Targeted Anticancer Agents.


Journal

Scientific reports
ISSN: 2045-2322
Titre abrégé: Sci Rep
Pays: England
ID NLM: 101563288

Informations de publication

Date de publication:
20 12 2019
Historique:
received: 05 06 2019
accepted: 19 11 2019
entrez: 22 12 2019
pubmed: 22 12 2019
medline: 11 11 2020
Statut: epublish

Résumé

In present investigation, an attempt was undertaken to modify the C-9 position of noscapine (Nos), an opium alkaloid to yield 9 -hydroxy methyl and 9 -carbaldehyde oxime analogues for augmenting anticancer potential. The synthesis of 9-hydroxy methyl analogue of Nos was carried out by Blanc reaction and 9-carbaldehyde oxime was engineered by oxime formation method and characterized using FT-IR,

Identifiants

pubmed: 31862933
doi: 10.1038/s41598-019-55839-8
pii: 10.1038/s41598-019-55839-8
pmc: PMC6925231
doi:

Substances chimiques

Antineoplastic Agents 0
Oximes 0
Noscapine 8V32U4AOQU

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

19542

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Auteurs

Vartika Tomar (V)

Department of Chemistry, University of Delhi, Delhi, 110007, India.
BioMedical Engineering Department, Faculty of Medicine, McGill University, Montreal, Canada.

Neeraj Kumar (N)

Department of Chemistry, University of Delhi, Delhi, 110007, India.

Ravi Tomar (R)

Department of Chemistry, University of Delhi, Delhi, 110007, India.

Damini Sood (D)

Department of Chemistry, University of Delhi, Delhi, 110007, India.

Neerupma Dhiman (N)

Amity Institute of Pharmacy, Noida, U.P, India.

Sujata K Dass (SK)

BL Kapur Hospital, New Delhi, 110005, India.

Satya Prakash (S)

BioMedical Engineering Department, Faculty of Medicine, McGill University, Montreal, Canada.

Jitender Madan (J)

Chandigarh College of Pharmacy, Mohali, Panjab, India.

Ramesh Chandra (R)

Department of Chemistry, University of Delhi, Delhi, 110007, India. acbrdu@hotmail.com.
Dr. B. R. Ambedkar Center for Biomedical Research, University of Delhi, Delhi, 110007, India. acbrdu@hotmail.com.

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Classifications MeSH