Roger L Papke

Affiliations

Department of Pharmacology and Therapeutics, College of Medicine (L.W.C., C.S., R.L.P.) and Department of Pharmacodynamics, College of Pharmacy, (J.L.W., L.R.M.), University of Florida, Gainesville, Florida; and Center for Drug Discovery, Research Triangle Institute, Durham, North Carolina (F.I.C.) rlpapke@ufl.edu.

Publications (30)

Nicotinic Acetylcholine Receptor Accessory Subunits Determine the Activity Profile of Epibatidine Derivatives.

Molecular pharmacology

Avec: Lu Wenchi Corrie , Clare Stokes , Jenny L Wilkerson , F Ivy Carroll , Lance R McMahon ,

Stable desensitization of α

European journal of pharmacology

Avec: Maria Chiara Pismataro , Nicole A Horenstein , Clare Stokes , Clelia Dallanoce , Ganesh A Thakur ,

Allosterically Potentiated

Molecular pharmacology

Avec: Douglas R Miller , Habibeh Khoshbouei , Sumanta Garai , Lucas N Cantwell , Clare Stokes , Ganesh Thakur ,

Selective Agonists and Antagonists of α9 Versus α7 Nicotinic Acetylcholine Receptors.

ACS chemical neuroscience

Avec: Hina Andleeb , Clare Stokes , Marta Quadri , Nicole A Horenstein

Silent agonists for α7 nicotinic acetylcholine receptors.

Pharmacological research

Avec: Marta Quadri , Alican Gulsevin

Synthesis, Pharmacological Characterization, and Structure-Activity Relationships of Noncanonical Selective Agonists for α7 nAChRs.

Journal of medicinal chemistry

Avec: Gisela Andrea Camacho-Hernandez , Clare Stokes , Brendan M Duggan , Katarzyna Kaczanowska , Stefania Brandao-Araiza , Lisa Doan , Palmer Taylor

A silent agonist of α7 nicotinic acetylcholine receptors modulates inflammation ex vivo and attenuates EAE.

Brain, behavior, and immunity

Avec: Jean-Rémi Godin , Patrick Roy , Marta Quadri , Deniz Bagdas , Wisam Toma , Ramya Narendrula-Kotha , Osama A Kishta , M Imad Damaj , Nicole A Horenstein , Alain R Simard

Nicotinic acetylcholine receptors: Conventional and unconventional ligands and signaling.

Neuropharmacology

Avec: Jon M Lindstrom

Therapeutic Targeting of

Pharmacological reviews

Avec: Nicole A Horenstein

The many enigmas of nicotine.

Advances in pharmacology (San Diego, Calif.)

Avec:

Betel quid: New insights into an ancient addiction.

Addiction biology

Avec: Clare Stokes , Jose A Pino , D Walker Hagan , Gonzalo E Torres , Edward A Phelps , Nicole A Horenstein ,

Cholinergic Receptors and Addiction.

Current topics in behavioral neurosciences

Avec: Darlene H Brunzell , Mariella De Biasi

The α7 nicotinic receptor silent agonist R-47 prevents and reverses paclitaxel-induced peripheral neuropathy in mice without tolerance or altering nicotine reward and withdrawal.

Experimental neurology

Avec: Wisam Toma , S Lauren Kyte , Deniz Bagdas , Asti Jackson , Julie A Meade , Faria Rahman , Zhi-Jian Chen , Egidio Del Fabbro , Lucas Cantwell , Abhijit Kulkarni , Ganesh A Thakur , John W Bigbee , David A Gewirtz , M Imad Damaj

Impact of modulation of the α7 nicotinic acetylcholine receptor on nicotine reward in the mouse conditioned place preference test.

Psychopharmacology

Avec: Asti Jackson , Y Alkhlaif , R L Papke , D H Brunzell , M I Damaj

The Allosteric Activation of α7 nAChR by α-Conotoxin MrIC Is Modified by Mutations at the Vestibular Site.

Toxins

Avec: Alican Gulsevin , Clare Stokes , Hue N T Tran , Aihua H Jin , Irina Vetter , Jens Meiler

Coffee and cigarettes: Modulation of high and low sensitivity α4β2 nicotinic acetylcholine receptors by n-MP, a biomarker of coffee consumption.

Neuropharmacology

Avec: Madison Karaffa , Nicole A Horenstein , Clare Stokes

Insights Into the Differential Desensitization of

Molecular pharmacology

Avec: Clare Stokes

Functions and pharmacology of α2β2 nicotinic acetylcholine receptors; in and out of the shadow of α4β2 nicotinic acetylcholine receptors.

Biochemical pharmacology

Avec:

Macroscopic and Microscopic Activation of

Molecular pharmacology

Avec: Marta Quadri , Sumanta Garai , Ganesh A Thakur , Clare Stokes , Alican Gulsevin , Nicole A Horenstein ,

Allosteric Agonism of

Molecular pharmacology

Avec: Alican Gulsevin , Clare Stokes , Sumanta Garai , Ganesh A Thakur , Marta Quadri , Nicole A Horenstein

Heteromeric Neuronal Nicotinic Acetylcholine Receptors with Mutant

The Journal of pharmacology and experimental therapeutics

Avec: Clare Stokes , Sumanta Garai , Abhijit R Kulkarni , Lucas N Cantwell , Colleen M Noviello , Ryan E Hibbs , Nicole A Horenstein , Khalil A Abboud , Ganesh A Thakur ,

In Silico Modeling of the α7 Nicotinic Acetylcholine Receptor: New Pharmacological Challenges Associated with Multiple Modes of Signaling.

Mini reviews in medicinal chemistry

Avec: Alican Gulsevin , Nicole Horenstein

Differing Activity Profiles of the Stereoisomers of 2,3,5,6TMP-TQS, a Putative Silent Allosteric Modulator of

Molecular pharmacology

Avec: Sumanta Garai , Clare Stokes , Nicole A Horenstein , Arthur D Zimmerman , Khalil A Abboud , Ganesh A Thakur

Effects of α7 Nicotinic Acetylcholine Receptor Positive Allosteric Modulator on BDNF, NKCC1 and KCC2 Expression in the Hippocampus following Lipopolysaccharide-Induced Allodynia and Hyperalgesia in a Mouse Model of Inflammatory Pain.

CNS & neurological disorders drug targets

Avec: Muzaffar Abbas , Sami Alzarea , Shafiqur Rahman

New Alpha9 nAChR Ligands Based on a 5-(Quinuclidin-3-ylmethyl)-1,2,4-oxadiazole Scaffold.

ACS chemical neuroscience

Avec: Clelia Dallanoce , Katrin Richter , Clare Stokes , Claudio Papotto , Hina Andleeb , Ganesh A Thakur , Andrew Kerr , Veronika Grau ,

Pharmacological characterization of 5-iodo-A-85380, a β2-selective nicotinic receptor agonist, in mice.

Journal of psychopharmacology (Oxford, England)

Avec: Lois S Akinola , Deniz Bagdas , Yasmin Alkhlaif , Asti Jackson , Cenk O Gurdap , Elnaz Rahimpour , F Ivy Carroll , M Imad Damaj

Pharmacological profiles and anti-inflammatory activity of pCN-diEPP and mCN-diEPP, new alpha9alpha10 nicotinic receptor ligands.

Neuropharmacology

Avec: Katrin Richter , Sara M Herz , Clare Stokes , M Imad Damaj , Veronika Grau ,

Design, synthesis, and electrophysiological evaluation of NS6740 derivatives: Exploration of the structure-activity relationship for alpha7 nicotinic acetylcholine receptor silent activation.

European journal of medicinal chemistry

Avec: Maria Chiara Pismataro , Nicole A Horenstein , Clare Stokes , Marta Quadri , Marco De Amici , Clelia Dallanoce

Cracking the Betel Nut: Cholinergic Activity of Areca Alkaloids and Related Compounds.

Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco

Avec: Nicole A Horenstein , Marta Quadri , Clare Stokes , Mohammed Shoaib ,

The α7 nicotinic acetylcholine receptor positive allosteric modulator prevents lipopolysaccharide-induced allodynia, hyperalgesia and TNF-α in the hippocampus in mice.

Pharmacological reports : PR

Avec: Muzaffar Abbas , Sami Alzarea , Shafiqur Rahman

Réseau de co-auteurs

Clare Stokes 17 collaborations

Nicole A Horenstein 12 collaborations

Ganesh A Thakur 7 collaborations

Marta Quadri 7 collaborations

Sumanta Garai 5 collaborations

Alican Gulsevin 5 collaborations

M Imad Damaj 4 collaborations

Clelia Dallanoce 3 collaborations

Deniz Bagdas 3 collaborations

Asti Jackson 3 collaborations

F Ivy Carroll 2 collaborations

Maria Chiara Pismataro 2 collaborations

Lucas N Cantwell 2 collaborations

Hina Andleeb 2 collaborations

Wisam Toma 2 collaborations

Khalil A Abboud 2 collaborations

Muzaffar Abbas 2 collaborations

Sami Alzarea 2 collaborations

Shafiqur Rahman 2 collaborations

Katrin Richter 2 collaborations

Veronika Grau 2 collaborations

Lu Wenchi Corrie 1 collaboration

Jenny L Wilkerson 1 collaboration

Lance R McMahon 1 collaboration

Douglas R Miller 1 collaboration

Habibeh Khoshbouei 1 collaboration

Ganesh Thakur 1 collaboration

Gisela Andrea Camacho-Hernandez 1 collaboration

Brendan M Duggan 1 collaboration

Katarzyna Kaczanowska 1 collaboration

Stefania Brandao-Araiza 1 collaboration

Lisa Doan 1 collaboration

Palmer Taylor 1 collaboration

Jean-Rémi Godin 1 collaboration

Patrick Roy 1 collaboration

Ramya Narendrula-Kotha 1 collaboration

Osama A Kishta 1 collaboration

Alain R Simard 1 collaboration

Jon M Lindstrom 1 collaboration

Jose A Pino 1 collaboration

D Walker Hagan 1 collaboration

Gonzalo E Torres 1 collaboration

Edward A Phelps 1 collaboration

Darlene H Brunzell 1 collaboration

Mariella De Biasi 1 collaboration

S Lauren Kyte 1 collaboration

Julie A Meade 1 collaboration

Faria Rahman 1 collaboration

Zhi-Jian Chen 1 collaboration

Egidio Del Fabbro 1 collaboration

Lucas Cantwell 1 collaboration

Abhijit Kulkarni 1 collaboration

John W Bigbee 1 collaboration

David A Gewirtz 1 collaboration

Y Alkhlaif 1 collaboration

R L Papke 1 collaboration

D H Brunzell 1 collaboration

M I Damaj 1 collaboration

Hue N T Tran 1 collaboration

Aihua H Jin 1 collaboration

Irina Vetter 1 collaboration

Jens Meiler 1 collaboration

Madison Karaffa 1 collaboration

Abhijit R Kulkarni 1 collaboration

Colleen M Noviello 1 collaboration

Ryan E Hibbs 1 collaboration

Nicole Horenstein 1 collaboration

Arthur D Zimmerman 1 collaboration

Claudio Papotto 1 collaboration

Andrew Kerr 1 collaboration

Lois S Akinola 1 collaboration

Yasmin Alkhlaif 1 collaboration

Cenk O Gurdap 1 collaboration

Elnaz Rahimpour 1 collaboration

Sara M Herz 1 collaboration

Marco De Amici 1 collaboration

Mohammed Shoaib 1 collaboration