Accueil
Klaus P Hoeflich
Klaus P Hoeflich
Affiliations
Blueprint Medicines, Cambridge, Massachusetts.
Publications (6)
Protein Kinase A Downregulation Delays the Development and Progression of Polycystic Kidney Disease.
Journal of the American Society of Nephrology : JASN
Avec:
Xiaofang Wang
,
Li Jiang
,
Ka Thao
,
Caroline R Sussman
,
Timothy LaBranche
,
Michael Palmer
,
Peter C Harris
,
G Stanley McKnight
,
Stefanie Schalm
,
Vicente E Torres
Machine Learning ADME Models in Practice: Four Guidelines from a Successful Lead Optimization Case Study.
ACS medicinal chemistry letters
Avec:
Alexander S Rich
,
Yvonne H Chan
,
Benjamin Birnbaum
,
Kamran Haider
,
Joshua Haimson
,
Michael Hale
,
Yongxin Han
,
William Hickman
,
Daniel Ortwine
,
Ayşegül Özen
,
David B Belanger
Evaluation of Protein Kinase cAMP-Activated Catalytic Subunit Alpha as a Therapeutic Target for Fibrolamellar Carcinoma.
Gastro hep advances
Avec:
Stefanie S Schalm
,
Erin O'Hearn
,
Kevin Wilson
,
Timothy P LaBranche
,
Grace Silva
,
Zhuo Zhang
,
Lucian DiPietro
,
Neil Bifulco
,
Richard Woessner
,
Nicolas Stransky
,
Darshan Sappal
,
Robert Campbell
,
Riadh Lobbardi
,
Michael Palmer
,
Joseph Kim
,
Chaoyang Ye
,
Marion Dorsch
,
Christoph Lengauer
,
Timothy Guzi
,
Vivek Kadambi
,
Andrew Garner
,
Acquired On-Target Clinical Resistance Validates FGFR4 as a Driver of Hepatocellular Carcinoma.
Cancer discovery
Avec:
Megan A Hatlen
,
Oleg Schmidt-Kittler
,
Cori Ann Sherwin
,
Emily Rozsahegyi
,
Nooreen Rubin
,
Michael P Sheets
,
Joseph L Kim
,
Chandrasekhar Miduturu
,
Neil Bifulco
,
Natasja Brooijmans
,
Hongliang Shi
,
Timothy Guzi
,
Andy Boral
,
Christoph Lengauer
,
Marion Dorsch
,
Richard D Kim
,
Yoon-Koo Kang
,
Beni B Wolf
,
First-in-Human Phase I Study of Fisogatinib (BLU-554) Validates Aberrant FGF19 Signaling as a Driver Event in Hepatocellular Carcinoma.
Cancer discovery
Avec:
Richard D Kim
,
Debashis Sarker
,
Tim Meyer
,
Thomas Yau
,
Teresa Macarulla
,
Joong-Won Park
,
Su Pin Choo
,
Antoine Hollebecque
,
Max W Sung
,
Ho-Yeong Lim
,
Vincenzo Mazzaferro
,
Joerg Trojan
,
Andrew X Zhu
,
Jung-Hwan Yoon
,
Sunil Sharma
,
Zhong-Zhe Lin
,
Stephen L Chan
,
Sandrine Faivre
,
Lynn G Feun
,
Chia-Jui Yen
,
Jean-Francois Dufour
,
Daniel H Palmer
,
Josep M Llovet
,
Melissa Manoogian
,
Meera Tugnait
,
Nicolas Stransky
,
Margit Hagel
,
Nancy E Kohl
,
Christoph Lengauer
,
Cori Ann Sherwin
,
Oleg Schmidt-Kittler
,
Hongliang Shi
,
Beni B Wolf
,
Yoon-Koo Kang
The pan-RAF-MEK non degrading molecular glue NST-628 is a potent and brain penetrant inhibitor of the RAS-MAPK pathway with activity across diverse RAS- and RAF-driven cancers.
Cancer discovery
Avec:
Meagan B Ryan
,
Bradley Quade
,
Natasha Schenk
,
Zhong Fang
,
Marshall Zingg
,
Steven E Cohen
,
Brooke M Swalm
,
Chun Li
,
Aysegul Ozen
,
Chaoyang Ye
,
Maria Stella Ritorto
,
Xin Huang
,
Arvin C Dar
,
Yongxin Han
,
Michael Hale
,
Margit Hagel
Réseau de co-auteurs
Christoph Lengauer
3 collaborations
Michael Palmer
2 collaborations
Michael Hale
2 collaborations
Yongxin Han
2 collaborations
Neil Bifulco
2 collaborations
Nicolas Stransky
2 collaborations
Chaoyang Ye
2 collaborations
Marion Dorsch
2 collaborations
Timothy Guzi
2 collaborations
Oleg Schmidt-Kittler
2 collaborations
Cori Ann Sherwin
2 collaborations
Hongliang Shi
2 collaborations
Richard D Kim
2 collaborations
Yoon-Koo Kang
2 collaborations
Beni B Wolf
2 collaborations
Margit Hagel
2 collaborations
Xiaofang Wang
1 collaboration
Li Jiang
1 collaboration
Ka Thao
1 collaboration
Caroline R Sussman
1 collaboration
Timothy LaBranche
1 collaboration
Peter C Harris
1 collaboration
G Stanley McKnight
1 collaboration
Stefanie Schalm
1 collaboration
Vicente E Torres
1 collaboration
Alexander S Rich
1 collaboration
Yvonne H Chan
1 collaboration
Benjamin Birnbaum
1 collaboration
Kamran Haider
1 collaboration
Joshua Haimson
1 collaboration
William Hickman
1 collaboration
Daniel Ortwine
1 collaboration
Ayşegül Özen
1 collaboration
David B Belanger
1 collaboration
Stefanie S Schalm
1 collaboration
Erin O'Hearn
1 collaboration
Kevin Wilson
1 collaboration
Timothy P LaBranche
1 collaboration
Grace Silva
1 collaboration
Zhuo Zhang
1 collaboration
Lucian DiPietro
1 collaboration
Richard Woessner
1 collaboration
Darshan Sappal
1 collaboration
Robert Campbell
1 collaboration
Riadh Lobbardi
1 collaboration
Joseph Kim
1 collaboration
Vivek Kadambi
1 collaboration
Andrew Garner
1 collaboration
Megan A Hatlen
1 collaboration
Emily Rozsahegyi
1 collaboration
Nooreen Rubin
1 collaboration
Michael P Sheets
1 collaboration
Joseph L Kim
1 collaboration
Chandrasekhar Miduturu
1 collaboration
Natasja Brooijmans
1 collaboration
Andy Boral
1 collaboration
Debashis Sarker
1 collaboration
Tim Meyer
1 collaboration
Thomas Yau
1 collaboration
Teresa Macarulla
1 collaboration
Joong-Won Park
1 collaboration
Su Pin Choo
1 collaboration
Antoine Hollebecque
1 collaboration
Max W Sung
1 collaboration
Ho-Yeong Lim
1 collaboration
Vincenzo Mazzaferro
1 collaboration
Joerg Trojan
1 collaboration
Andrew X Zhu
1 collaboration
Jung-Hwan Yoon
1 collaboration
Sunil Sharma
1 collaboration
Zhong-Zhe Lin
1 collaboration
Stephen L Chan
1 collaboration
Sandrine Faivre
1 collaboration
Lynn G Feun
1 collaboration
Chia-Jui Yen
1 collaboration
Jean-Francois Dufour
1 collaboration
Daniel H Palmer
1 collaboration
Josep M Llovet
1 collaboration
Melissa Manoogian
1 collaboration
Meera Tugnait
1 collaboration
Nancy E Kohl
1 collaboration
Meagan B Ryan
1 collaboration
Bradley Quade
1 collaboration
Natasha Schenk
1 collaboration
Zhong Fang
1 collaboration
Marshall Zingg
1 collaboration
Steven E Cohen
1 collaboration
Brooke M Swalm
1 collaboration
Chun Li
1 collaboration
Aysegul Ozen
1 collaboration
Maria Stella Ritorto
1 collaboration
Xin Huang
1 collaboration
Arvin C Dar
1 collaboration