Repositioning Brusatol as a Transmission Blocker of Malaria Parasites.

brusatol drug discovery malaria natural products quassinoids transmission blocking

Journal

ACS infectious diseases
ISSN: 2373-8227
Titre abrégé: ACS Infect Dis
Pays: United States
ID NLM: 101654580

Informations de publication

Date de publication:
01 Oct 2024
Historique:
medline: 3 10 2024
pubmed: 3 10 2024
entrez: 1 10 2024
Statut: aheadofprint

Résumé

Currently, primaquine is the only malaria transmission-blocking drug recommended by the WHO. Recent efforts have highlighted the importance of discovering new agents that regulate malarial transmission, with particular interest in agents that can be administered in a single low dose, ideally with a discrete and

Identifiants

pubmed: 39352879
doi: 10.1021/acsinfecdis.4c00434
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Auteurs

Amelia Cox (A)

School of Biodiversity, One Health and Veterinary Medicine, College of Medical, Veterinary and Life Sciences, University of Glasgow, Garscube Campus, Bearsden Road, Glasgow G61 1QH, United Kingdom.

Neelima Krishnankutty (N)

Institute of Immunology and Infection Research, University of Edinburgh, Ashworth Laboratories 2, Room 3.11, Edinburgh EH9 3FL, United Kingdom.

Steven Shave (S)

School of Biological Sciences, University of Edinburgh, The King's Buildings, Edinburgh EH9 3BF, United Kingdom.

Virginia M Howick (VM)

School of Biodiversity, One Health and Veterinary Medicine, College of Medical, Veterinary and Life Sciences, University of Glasgow, Garscube Campus, Bearsden Road, Glasgow G61 1QH, United Kingdom.

Manfred Auer (M)

School of Biological Sciences, University of Edinburgh, The King's Buildings, Edinburgh EH9 3BF, United Kingdom.
Xenobe Research Institute, P.O. Box 3052, San Diego, California 92163, United States.

James J La Clair (JJ)

Xenobe Research Institute, P.O. Box 3052, San Diego, California 92163, United States.

Nisha Philip (N)

Institute of Immunology and Infection Research, University of Edinburgh, Ashworth Laboratories 2, Room 3.11, Edinburgh EH9 3FL, United Kingdom.

Classifications MeSH