Synthesis of ciprofloxacin-linked 1,2,3-triazole conjugates as potent antibacterial agents using click chemistry: exploring their function as DNA gyrase inhibitors


Journal

RSC advances
ISSN: 2046-2069
Titre abrégé: RSC Adv
Pays: England
ID NLM: 101581657

Informations de publication

Date de publication:
22 May 2024
Historique:
received: 21 02 2024
accepted: 11 05 2024
medline: 31 5 2024
pubmed: 31 5 2024
entrez: 31 5 2024
Statut: epublish

Résumé

The antibacterial efficacy of some newly developed C-3 carboxylic group-containing ciprofloxacin-linked 1,2,3-triazole conjugates was studied. Twenty-one compounds from three different series of triazoles were synthesized using click chemistry and evaluated for their antibacterial activity against nine different pathogenic strains, including three Gram-positive strains,

Identifiants

pubmed: 38818013
doi: 10.1039/d4ra01332h
pii: d4ra01332h
pmc: PMC11138863
doi:

Types de publication

Journal Article

Langues

eng

Pagination

17051-17070

Informations de copyright

This journal is © The Royal Society of Chemistry.

Déclaration de conflit d'intérêts

The authors have no conflict of Interest for manuscript publication.

Auteurs

Upendra Kumar Patel (UK)

Department of Medicinal Chemistry, Institute of Medical Sciences, Banaras Hindu University Varanasi UP-221005 India agarwal.dralka@gmail.com.

Punit Tiwari (P)

Department of Microbiology, Institute of Medical Sciences, Banaras Hindu University Varanasi UP-221005 India.

Ragini Tilak (R)

Department of Microbiology, Institute of Medical Sciences, Banaras Hindu University Varanasi UP-221005 India.

Gaurav Joshi (G)

Department of Pharmaceutical Sciences, Hemvati Nandan Bahuguna Garhwal University (Central University) Dist. Garhwal (Uttarakhand) Srinagar-246174 India.

Roshan Kumar (R)

Department of Microbiology, Central University of Punjab Ghudda Bathinda-151401 India.

Alka Agarwal (A)

Department of Medicinal Chemistry, Institute of Medical Sciences, Banaras Hindu University Varanasi UP-221005 India agarwal.dralka@gmail.com.

Classifications MeSH