Galantamine Based Novel Acetylcholinesterase Enzyme Inhibitors: A Molecular Modeling Design Approach.
ADME
Alzheimer’s disease
molecular docking and molecular dynamics
Journal
Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009
Informations de publication
Date de publication:
19 Jan 2023
19 Jan 2023
Historique:
received:
01
10
2022
revised:
31
12
2022
accepted:
09
01
2023
entrez:
11
2
2023
pubmed:
12
2
2023
medline:
15
2
2023
Statut:
epublish
Résumé
Acetylcholinesterase (AChE) enzymes play an essential role in the development of Alzheimer's disease (AD). Its excessive activity causes several neuronal problems, particularly psychopathies and neuronal cell death. A bioactive pose on the
Identifiants
pubmed: 36770702
pii: molecules28031035
doi: 10.3390/molecules28031035
pmc: PMC9919016
pii:
doi:
Substances chimiques
Cholinesterase Inhibitors
0
Galantamine
0D3Q044KCA
Acetylcholinesterase
EC 3.1.1.7
Enzyme Inhibitors
0
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Références
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