Development of a multigram synthesis of the bradykinin receptor 2 agonist FR-190997 and analogs thereof.
B2R agonists
FR-190997
cancer
late-stage diversification
quinolines
Journal
Archiv der Pharmazie
ISSN: 1521-4184
Titre abrégé: Arch Pharm (Weinheim)
Pays: Germany
ID NLM: 0330167
Informations de publication
Date de publication:
May 2023
May 2023
Historique:
revised:
24
12
2022
received:
28
11
2022
accepted:
13
01
2023
medline:
8
5
2023
pubmed:
1
2
2023
entrez:
31
1
2023
Statut:
ppublish
Résumé
Using Fujisawa's B2R agonist FR-190997, we recently demonstrated for the first time that agonism at the bradykinin receptor type 2 (B2R) produces substantial antiproliferative effects. FR-190997 elicited an EC
Identifiants
pubmed: 36720040
doi: 10.1002/ardp.202200610
doi:
Substances chimiques
FR 190997
0
Receptor, Bradykinin B2
0
Quinolines
0
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Pagination
e2200610Informations de copyright
© 2023 Deutsche Pharmazeutische Gesellschaft.
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