Simulating the Hydrodynamic Conditions of the Human Ascending Colon: A Digital Twin of the Dynamic Colon Model.

Dynamic Colon Model (DCM) Magnetic Resonance Imaging (MRI) Smoothed Particle Hydrodynamics (SPH) colon colon targeted drug delivery digital twin discrete multiphysics dissolution apparatus large intestine shear rate

Journal

Pharmaceutics
ISSN: 1999-4923
Titre abrégé: Pharmaceutics
Pays: Switzerland
ID NLM: 101534003

Informations de publication

Date de publication:
13 Jan 2022
Historique:
received: 09 12 2021
revised: 26 12 2021
accepted: 11 01 2022
entrez: 21 1 2022
pubmed: 22 1 2022
medline: 22 1 2022
Statut: epublish

Résumé

The performance of solid oral dosage forms targeting the colon is typically evaluated using standardised pharmacopeial dissolution apparatuses. However, these fail to replicate colonic hydrodynamics. This study develops a digital twin of the Dynamic Colon Model; a physiologically representative in vitro model of the human proximal colon. Magnetic resonance imaging of the Dynamic Colon Model verified that the digital twin robustly replicated flow patterns under different physiological conditions (media viscosity, volume, and peristaltic wave speed). During local contractile activity, antegrade flows of 0.06-0.78 cm s

Identifiants

pubmed: 35057077
pii: pharmaceutics14010184
doi: 10.3390/pharmaceutics14010184
pmc: PMC8778200
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : Medical Research Council
ID : MC_PC_18040
Pays : United Kingdom
Organisme : EPSRC Centre for Doctoral Training in Formulation Engineering
ID : EP/L015153/1
Organisme : Engineering and Physical Sciences Research Council
ID : EP/S019227/1

Commentaires et corrections

Type : ErratumIn

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Auteurs

Michael Schütt (M)

School of Chemical Engineering, University of Birmingham, Edgbaston, Birmingham B15 2TT, UK.

Connor O'Farrell (C)

School of Chemical Engineering, University of Birmingham, Edgbaston, Birmingham B15 2TT, UK.

Konstantinos Stamatopoulos (K)

School of Chemical Engineering, University of Birmingham, Edgbaston, Birmingham B15 2TT, UK.
Biopharmaceutics, Pharmaceutical Development, PDS, MST, RD Platform Technology & Science, GSK, David Jack Centre, Park Road, Ware, Hertfordshire SG12 0DP, UK.

Caroline L Hoad (CL)

Nottingham Digestive Diseases Centre and National Institute for Health Research (NIHR) Nottingham Biomedical Research Centre, Nottingham University Hospitals NHS Trust and University of Nottingham, Nottingham NG7 2UK, UK.
Sir Peter Mansfield Imaging Centre, School of Physics and Astronomy, University of Nottingham, Nottingham NG7 2RD, UK.

Luca Marciani (L)

Nottingham Digestive Diseases Centre and National Institute for Health Research (NIHR) Nottingham Biomedical Research Centre, Nottingham University Hospitals NHS Trust and University of Nottingham, Nottingham NG7 2UK, UK.

Sarah Sulaiman (S)

Nottingham Digestive Diseases Centre and National Institute for Health Research (NIHR) Nottingham Biomedical Research Centre, Nottingham University Hospitals NHS Trust and University of Nottingham, Nottingham NG7 2UK, UK.

Mark J H Simmons (MJH)

School of Chemical Engineering, University of Birmingham, Edgbaston, Birmingham B15 2TT, UK.

Hannah K Batchelor (HK)

Strathclyde Institute of Pharmacy and Biomedical Sciences, University of Strathclyde, 161 Cathedral Street, Glasgow G4 0RE, UK.

Alessio Alexiadis (A)

School of Chemical Engineering, University of Birmingham, Edgbaston, Birmingham B15 2TT, UK.

Classifications MeSH