Sustainable Triazine-Based Dehydro-Condensation Agents for Amide Synthesis.


Journal

Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009

Informations de publication

Date de publication:
02 Jan 2021
Historique:
received: 08 12 2020
revised: 22 12 2020
accepted: 29 12 2020
entrez: 6 1 2021
pubmed: 7 1 2021
medline: 4 9 2021
Statut: epublish

Résumé

Conventional methods employed today for the synthesis of amides often lack of economic and environmental sustainability. Triazine-derived quaternary ammonium salts, e.g., 4-(4,6-dimethoxy-1,3,5-triazin-2-yl)-4-methylmorpholinium chloride (DMTMM(Cl)), emerged as promising dehydro-condensation agents for amide synthesis, although suffering of limited stability and high costs. In the present work, a simple protocol for the synthesis of amides mediated by 2-chloro-4,6-dimethoxy-1,3,5-triazine (CDMT) and a

Identifiants

pubmed: 33401732
pii: molecules26010191
doi: 10.3390/molecules26010191
pmc: PMC7795458
pii:
doi:

Substances chimiques

Amides 0
Amines 0
Benzamides 0
Carboxylic Acids 0
N-phenethylbenzamide 0
Perchlorates 0
Phenethylamines 0
Piperazines 0
Quaternary Ammonium Compounds 0
Solvents 0
Triazines 0
1,4-dimethylpiperazine TF146U602L
perchlorate VLA4NZX2P4

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

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Auteurs

Roberto Sole (R)

Dipartimento di Scienze Molecolari e Nanosistemi, Università Ca' Foscari di Venezia, Via Torino 155, 30172 Venezia, Italy.

Vanessa Gatto (V)

Crossing srl, Viale della Repubblica 193/b, 31100 Treviso, Italy.

Silvia Conca (S)

Dipartimento di Scienze Molecolari e Nanosistemi, Università Ca' Foscari di Venezia, Via Torino 155, 30172 Venezia, Italy.

Noemi Bardella (N)

Dipartimento di Scienze Molecolari e Nanosistemi, Università Ca' Foscari di Venezia, Via Torino 155, 30172 Venezia, Italy.

Andrea Morandini (A)

Dipartimento di Scienze Molecolari e Nanosistemi, Università Ca' Foscari di Venezia, Via Torino 155, 30172 Venezia, Italy.

Valentina Beghetto (V)

Dipartimento di Scienze Molecolari e Nanosistemi, Università Ca' Foscari di Venezia, Via Torino 155, 30172 Venezia, Italy.
Crossing srl, Viale della Repubblica 193/b, 31100 Treviso, Italy.

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Classifications MeSH