Structure-Activity Relationship Studies of α-Ketoamides as Inhibitors of the Phospholipase A and Acyltransferase Enzyme Family.
Journal
Journal of medicinal chemistry
ISSN: 1520-4804
Titre abrégé: J Med Chem
Pays: United States
ID NLM: 9716531
Informations de publication
Date de publication:
10 09 2020
10 09 2020
Historique:
pubmed:
14
8
2020
medline:
15
12
2020
entrez:
14
8
2020
Statut:
ppublish
Résumé
The phospholipase A and acyltransferase (PLAAT) family of cysteine hydrolases consists of five members, which are involved in the Ca
Identifiants
pubmed: 32787138
doi: 10.1021/acs.jmedchem.0c00522
pmc: PMC7498158
doi:
Substances chimiques
Amides
0
Enzyme Inhibitors
0
Acyltransferases
EC 2.3.-
Phospholipases
EC 3.1.-
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
9340-9359Références
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